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EGFR exon 20 insertions (excluding A763_Y764insFQEA) are insensitive to classical EGFR-TK...

Deterministic view of the source YAML entity. Clinical authority remains with the cited source IDs and reviewer sign-off state.

IDBMA-EGFR-EX20INS-NSCLC
TypeActionability
Statusreviewed 2026-04-27 | pending_clinical_signoff | actionability review required
DiseasesDIS-NSCLC
SourcesSRC-CIVIC SRC-ESMO-NSCLC-METASTATIC-2024 SRC-NCCN-NSCLC-2025

Actionability Facts

BiomarkerBIO-EGFR-MUTATION
Variantexon 20 insertion
DiseaseDIS-NSCLC
ESCAT tierIA
Recommended combinationsamivantamab + carboplatin + pemetrexed (PAPILLON 1L), amivantamab monotherapy (2L), platinum-doublet chemotherapy (alternative)
Contraindicated monotherapyosimertinib (poor activity in classical ex20ins), gefitinib / erlotinib / afatinib (resistant), mobocertinib (withdrawn 2023-2024)
Evidence summaryEGFR exon 20 insertions (excluding A763_Y764insFQEA) are insensitive to classical EGFR-TKIs. Amivantamab (EGFR-MET bispecific) + chemo is 1L standard (PAPILLON, Zhou et al. 2023). Mobocertinib was withdrawn globally 2023-2024 for failed confirmatory trial. Sunvozertinib (China-approved) is an emerging option in 2L.

Notes

ESCAT IA per PAPILLON. OncoKB Level 1. NGS preferred over PCR for detection — many ex20ins variants missed by hotspot PCR panels. A763_Y764insFQEA is the rare classical-TKI-sensitive exception.

Used By

No reverse references found in the YAML corpus.