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Radium-223 dichloride

Deterministic view of the source YAML entity. Clinical authority remains with the cited source IDs and reviewer sign-off state.

IDDRUG-RADIUM-223
TypeDrug
Aliases
XofigoРадій-223 дихлорид
Statuspending_clinical_signoff
DiseasesDIS-PROSTATE
SourcesSRC-ESMO-PROSTATE-2024 SRC-NCCN-PROSTATE-2025

Drug Facts

ClassBone-seeking α-emitter
MechanismCalcium-mimetic α-emitter that incorporates into hydroxyapatite at sites of high bone turnover (osteoblastic metastases). α-radiation has ~100 µm range — high local tumor cell kill with minimal marrow toxicity vs β-emitters.
Typical dosing55 kBq/kg IV q4 weeks × 6 cycles. Symptomatic bone-predominant mCRPC without visceral metastases (visceral mets exclude — ALSYMPCA exclusion criterion).
Ukraine registeredTrue
NSZU reimbursedFalse
Ukraine last verified2026-04-27

Notes

ALSYMPCA: OS benefit + symptomatic skeletal-event reduction in bone-predominant mCRPC. ERA-223 caution: avoid combination with abiraterone (use sequentially). UA-access barrier.

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Regimens