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Momelotinib

Deterministic view of the source YAML entity. Clinical authority remains with the cited source IDs and reviewer sign-off state.

IDDRUG-MOMELOTINIB
TypeDrug
Aliases
OjjaaraOmjjaraМомелотиніб
Statusreviewed 2026-04-25 | pending_clinical_signoff
DiseasesDIS-PMF
SourcesSRC-COMFORT-I-VERSTOVSEK-2012 SRC-NCCN-MPN-2025

Drug Facts

ClassJAK1/JAK2 + ACVR1 inhibitor
MechanismJAK1/JAK2 inhibitor with additional ACVR1 inhibition that lowers hepcidin → improves anemia. Distinguishes momelotinib from ruxolitinib (which often worsens anemia). 2L for MF with anemia.
Typical dosingMF: 200 mg PO once daily with or without food. Renal/hepatic dose adjustments apply.
Ukraine registeredFalse
NSZU reimbursedFalse
Ukraine last verified2026-04-27

Notes

Approved for MF with anemia (Hb <10) — MOMENTUM trial: spleen response + symptom improvement + Hb improvement compared with danazol. NOT registered in Ukraine. HBV / TB screening required before initiation.

Used By

Regimens