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Lutetium-177 PSMA-617

Deterministic view of the source YAML entity. Clinical authority remains with the cited source IDs and reviewer sign-off state.

IDDRUG-LUTETIUM-177-PSMA
TypeDrug
Aliases
PluvictoЛютецій-177 PSMA-617
Statuspending_clinical_signoff
DiseasesDIS-PROSTATE
SourcesSRC-ESMO-PROSTATE-2024 SRC-NCCN-PROSTATE-2025

Drug Facts

ClassPSMA-targeted radioligand (β-emitter)
MechanismSmall-molecule PSMA-binding ligand conjugated to β-emitting radionuclide Lu-177. PSMA is expressed on >90% of prostate adenocarcinoma cells; Lu-177-PSMA-617 binds PSMA and delivers cytotoxic β-radiation directly to tumor sites. Requires PSMA-PET-positive disease for selection (VISION criteria).
Typical dosing7.4 GBq IV q6 weeks × 6 cycles (VISION protocol). Administered in nuclear medicine / radioligand therapy unit with appropriate radiation safety.
Ukraine registeredFalse
NSZU reimbursedFalse
Ukraine last verified2026-04-27

Notes

VISION trial: significant rPFS + OS benefit in PSMA-PET-positive mCRPC post-ARPI + post-taxane. Requires nuclear medicine infrastructure + PSMA-PET availability — limits access in Ukraine to a few centers.

Used By

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Regimens